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Ana Sayfa Yağlar Enzimler Mineraller Proteinler Vitaminler Nükleik Asitler Karbonhidratlar Hormonlar Temel Biyokimya Makaleler

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Ana Sayfa
Carcinogenesis/Mutagenesis PDF Yazdır
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Carcinogenesis/Mutagenesis

P29
Benzene hexachlorides induce TOP2A expression in human primary renal cells
Keiko Hosohata, School of Medicine, Jichi Medical University; Hitoshi Ando, School of Medicine, Jichi Medical University; Akira Sasaki, School of Medicine, Jichi Medical University; Yasuo Oshima, School of Medicine, Jichi Medical University; Akio Fujimura, School of Medicine, Jichi Medical University
P30
CYP2E1*5B Polymorphism, Response to Chemotherapy and Survival in Non Small Cell Lung Cancer Patients
Volkan Karacaoglan, Ankara University, Faculty of Pharmacy; Ahmet Oguz Ada, Ankara University, Faculty of Pharmacy; Semih C. Kunak, Giresun University, Medical Faculty; Sibel Alpar, Ataturk Pulmonary Diseases and Thoracic Surgery Hospital; Meral Gulhan, Ataturk Pulmonary Diseases and Thoracic Surgery Hospital; Bahar Kurt, Ataturk Pulmonary Diseases and Thoracic Surgery Hospital; Mumtaz Iscan, Ankara University, Faculty of Pharmacy
P31
Cytogenetical and Cytological EFFECTS of the Diclofenac IN PLANTS Test Systems
Rena Agabeyli, Institute of Botany, National Academy of Sciences
P32
Effect of DDT on the target genes of hormonal carcinogenesis
Vladimir Pustylnyak, Institute of MolBiol & Bioph SB RAMS; Mariya Liyasova, Institute of MolBiol and Bioph SB RAMS; Lyudmila F. Gulyaeva, Institute of MolBiol and Bioph SB RAMS
P33
Modification with Plant’S Product Xenobiotics Induced CHROMOSOMAL Instability IN the PLANTS and Anymals CELLS
Rena Agabeyli, Institute of Botany
P34
Predicting the Genotoxicity of Allylbenzene Compounds
Alex Cayley, Lhasa Limited; Richard Williams, Lhasa Limited
P35
Predictive Gene-expression Signatures of Non-Genotoxic Carcinogen Responses in Mouse Embryonic Stem Cells
Bob van de Water, LACDR, Leiden University; Ilse Huijskens, LACDR, Leiden University; Martijs Jonker, University of Amsterdam; Timo Breit, University of Amsterdam; Harry Vrieling, Leiden University Medical Center
P36
Who is most susceptible to arsenic-induced internal malignancies?
Ling-I Hsu, Academia Sinica
 
Biomarkers PDF Yazdır
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Biomarkers

P21
Biomarkers releated to endothelial dysfunction in the “peripheral arterial disease” (PAD)
Suzan E. Usanmaz, Ankara University, Faculty of Medicine; Cuneyt Koksoy, Ankara University, Faculty of Medicine; Emine Demirel-Yilmaz, Ankara University, Faculty of Medicine
P22
Comet Assay and Cytokinesis-Blocked Micronucleus Test for Monitoring The Genotoxic Effects of Narrowband UVB Treatment in Psoriasis Patients
Diren Beyoglu, Marmara University, Faculty of Pharmacy; Zehra Asiran Serdar, Haydarpasa Numune Training and Research Hospital; Ilkin Zindanci, Goztepe Training and Research Hospital; Gulden Z. Omurtag, Marmara University, Faculty of Pharmacy; Semra Sardas, Marmara University, Faculty of Pharmacy
P23
MALDI -Imaging of Endogenous Lipids in Tumour Xenographs
Philip Bond, Quotient Bioresearch Limited; Andrew B. McEwen, Quotient Bioresearch (Rushden) Limited; Stuart G. Wood, Quotient Bioresearch (Rushden) Limited; Malcolm Clench, Sheffield Hallam University
P24
Urinary excretion of the acrylonitrile metabolite 2-cyanoethylmercapturic acid is correlated with tobacco smoke exposure
Emmanuel Minet, British American Tobacco; Francis Cheung, British American Tobacco; Graham Errington, British American Tobacco; Katharina Sterz, Analytisch-Biologisches Forschungslabor GmbH; Gerhard Scherer, Analytisch-Biologisches Forschungslabor GmbH
 
Bioavailability PDF Yazdır
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Bioavailability

Analysis of Factors Determining Incomplete Intestinal Drug Absorption as Observed in Cyclosporine Formulations by Use of Tube Model Incorporated Nernst Equation
Katsumi Iga, Doshisha Women's College of Liberal Arts; Akiko Kiriyama, Doshisha Women's College of Liberal Arts; Akino Honbo, Doshisha Women's College of Liberal Arts
The Influence of Albumin to Brain Tissue Binding
Hinnerk Boriss, Sovicell GmbH; Lydia Helmdach, University of Halle
Poor Membrane Permeability Ability of SANT75 across Caco-2 Cell Monolayer Due to High Cellular Accumulation
Na Li, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Ying Hu, Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Yang Yu, Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Song Li, Shenzhen Graduate School of Peking University, Shenzhen, 518055, China; Chao Che, Shenzhen Biosynergo Bio Technology Co.,Ltd,Shenzhen, 518055, China; Ling Yang, Dalian Institute of Chemical Physics, Chinese Academy of Sciences
hCYP3A4 Over-Expressing IEC-18 Cell Lines as an In Vitro Model to Assess Gut Permeability and CYP3A4 Metabolism
Swathi Vangala, University of the Pacific; Jae H. Chang, Genentech; Ning Liu, Genentech; William K. Chan, Univ of the Pacific; Miki S. Park, Univ of Pacific
 
Cytochrome P450 PDF Yazdır
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Cytochrome P450

Assessment of Effects of IR and IPC on Activities of Cytochrome P450 Isoforms in Rats by a Five-Drug Cocktail Approach
Jianshi Lou, Tianjin Medical University; Ying Liu, Tianjin Medical University; Qin LI, Tianjin Medical University; Jianjie Jiao, Tianjin Medical University; Caili Zhang, Tianjin Medical University
Functional Characterization of Recombinant NADPH-P450 Reductase Protein from Candida albicans
Hyoung-Goo Park, Konkuk University; Young-Jin Chun, Chung-Ang University; Donghak Kim, Konkuk University
Expression and Inducibility by Phenobarbital of CYP2C33, CYP2C42 CYP2C49, CYP2B22 and CYP3As in Liver, Kidney, Small Intestine and Nasal Tissues of Pig
Emanuela Puccinelli, Institute of Clinical Physiology, CNR, via Moruzzi 1, 56100 Pisa, Italy; Pier Giovanni Gervasi, Institute of Clinical Physiology, CNR, via Moruzzi 1, 56100 Pisa, Italy; Margherita la Marca, Institute of Agricultural Biotechnology, CNR, via Moruzzi 1, 56100 Pisa, Italy; Pascale Beffy, Institute of Clinical Physiology, CNR, via Moruzzi 1, 56100 Pisa, Italy; Vincenzo Longo, Institute of Agricultural Biotechnology, CNR, via Moruzzi 1, 56100 Pisa, Italy
Absolute Quantification of CYP27A1 and CYP46A1 in the Human Brain and Retina
Illarion V. Turko, Center for Advanced Research in Biotechnology; Wei-Li Liao, Center for Advanced Research in Biotechnology; Gun-Young Heo, Case Western Reserve University; Rachel E. Reem, Case Western Reserve University; Nathan G. Dodder, National Institute of Standards and Technology; Pier Luigi DiPatre, University of Texas Medical Branch; Irina A. Pikuleva, Case Western Reserve University
Probabilistic GALAS Models For The Prediction Of The Human Cytochrome P450 Inhibition
Remigijus Didziapetris, ACD/Labs, Inc.; Justas Dapkunas, ACD/Labs, Inc.; Andrius Sazonovas, ACD/Labs, Inc.; Pranas Japertas, ACD/Labs, Inc.
Dexamethasone Enhances CYP3A-mediated Inactivation of Active Vitamin D3 Metabolite in Mouse Liver
Subrata Deb, Vancouver Prostate Centre; Mitali Pandey, Vancouver Prostate Centre; Hans Adomat, Vancouver Prostate Centre; Emma Guns, Vancouver Prostate Centre
Influence of CYP2C9 polymorphism on metabolism of Valproate and its hepatotoxin metabolite in Iranian patients
Abbas Kebriaeezadeh, Tahran University of Medical Sciences; Noushin amini-Shirazi, Tums
The inhibitory effect of quercetin on rat hepatal CYP2D2
Ondrej Zendulka, Masaryk University; Jan Jurica, Masaryk University; Alexandra Sulcova, Masaryk University
Humanized CYP3A Mice: (1) Construction of Humanized MODEL Mice CONTAINING the CYP3A Cluster for Drug Screening
Yasuhiro Kazuki, Tottori University; Satoshi Abe, Tottori University; Masato Takiguchi, Tottori University; Hidetoshi Hoshiya, Tottori University; Naoyo Kajitani, Tottori University; Toko Yoshino, Tottori University; Shoko Takehara, Tottori University; Chie Ishihara, Tottori University; Kinya Kubo, Tottori University; Takeshi Oshima, Inovative Drug Research Laboratories, Kyowa Hakko Kirin CO. Ltd; Kazuma Tomizuka, Inovative Drug Research Laboratories, Kyowa Hakko Kirin CO. Ltd; Sasitorn Aueviriyavit, Chiba Univestiry; Kaoru Kobayashi, Chiba Univestiry; Kan Chiba, Chiba Univestiry; Yasuko Tsukazaki, Mitsubishi Chemical Medience Corporation; Naoto Senda, Mitsubishi Chemical Medience Corporation; Mitsuo Oshimura, Tottori University
Humanized CYP3A mice : (3)Metabolism of CYP3A4 substrates detected by LC/MS system
Yasuko Tsukazaki, Mitsubishi Chemical Medience Corporation; Manabu Nishii, Mitsubishi Chemical Medience Corporation; Naoto Senda, Mitsubishi Chemical Medience Corporation; Kazuki Yasuhiro, Tottori University; Kinya Kubo, Tottori University; Kaoru Kobayashi, Chiba University; Kan Chiba, Chiba University; Shigeru Yamada, K. K. AB Sciex.; Tetsuo Kokaji, K. K. AB Sciex.; Masakazu Takahashi, GL Sciences Inc.; Hiroshi Igarashi, GL Sciences Inc.; Mitsuo Oshimura, Tottori University
CYP2E1 INDUCTION and Oxidative STRESS IN CEREBELLAR Granule Neurons
Ana Carolina Valencia-Olvera, Instituto de Investigaciones Biomédicas, Universidad Nacional Autónoma de México; Julio Morán, Instituto de Fisiología Celular, Universidad Nacional Autónoma de México; Rafael Camacho-Carranza, Instituto de Investigaciones Biomédicas, Universidad Nacional Autónoma de México; Jesús Javier Espinosa-Aguirre, Instituto de Investigaciones Biomédicas, Universidad Nacional Autónoma de México
Cryopreserved HUMAN Hepatocytes as A MODEL for the EVALUATION of TOXICITY and Drug-Drug Interactions
Lysiane Richert, KaLy-Cell; Audrey Baze, KaLy-Cell; Coraline Desbans, KaLy-Cell; Celine Parmentier, KaLy-Cell; Bruno Heyd, Service de Chirurgie Viscérale et Digestive; Georges Mantion, Service de Chirurgie Viscérale et Digestive; Philippe Bachellier, Centre de Chirurgie Viscérale et de Transplantation; Jean-Christophe Weber, Clinique de l'Orangerie; Thomas Zacharias, CHU Mulhouse; Sandrine Simon, F. Hoffmann-La Roche Ltd.; Anna-Lena Ungell, AstraZeneca R&D; Pieter Annaert, Katholieke Universiteit Leuven; Eliane Alexandre, KaLy-Cell
Bupropion Hydroxylation As A Selective Marker Of Rat Cytochrome P450 2B1 Catalytic Activity
Dumrongsak Pekthong, KaLy-Cell; Alexandre Bonet, Laboratoire de Toxicologie Cellulaire, EA 4267, IFR 133; Lysiane Richert, KaLy-Cell; Hélène Martin, Laboratoire de Toxicologie Cellulaire, EA 4267, IFR 133
Metabolic Ratio of Dextromethorphan/dextrorphan in CYP2D6 Phenotyping - Identification of Cut-off Values in Serum and Correlation With Urine Levels
Jan Jurica, Masaryk University, Faculty of Medicine; Ondrej Zendulka, Masaryk University, Faculty of Medicine; Richard Bartecek, Faculty Hospital Brno and Faculty of Medicine, Masaryk University; Alexandra Zourkova, Faculty Hospital Brno and Faculty of Medicine, Masaryk University; Eva Flodrova, Faculty Hospital Brno; Jana Zrustova, Faculty Hospital Brno; Alexandra Sulcova, Masaryk University
The “Albumin Effect” on In vitro Kinetics of Various Cytochrome P450-Catalyzed Reactions: In vitro to In vivo Extrapolation
Nitsupa Wattanachai, Faculty of Medicine, Khon Kaen University; Wichittra Tassaneeyakul, Faculty of Medicine, Khon Kaen University; Verawan Uchaipichat, Faculty of Pharmaceutical Sciences, Khon Kaen University; John O. Miners, Flinders University School of Medicine
A simple sampling strategy to assess activity of CYP3A in vivo using deoxyschizandrin as a probe
Jing-jing Wu, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Yan-Yan Zhang, Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Ying Hu, Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Si-Cheng Liang, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Ling Yang, Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences
Characterization of in vitro bioactivation of rutaecarpine in human liver microsomes (HLMs)
Zhong-Ze Fang, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Ling Yang, Dalian Institute of Chemical Physics, Chinese Academy of Sciences
Characterization of in vitro bioactivation of Noscapine in Human Liver Microsomes
Zhong-Ze Fang, Dalian Institute of Chemical Physics, Chinese Academy of Sciences; Ling Yang, Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences
Simultaneous Evaluation of Influence of Scutellaria Baicalensis Georgi on CYP450 by Cocktail Probe Drugs
Qin Li, Tianjin Medical University; Jianjie Jiao, Tianjin Medical University; Xiaowen Han, Tianjin Medical University; Jianshi Lou, Tianjin Medical University
Engineering Bacillus megaterium CYP102A1 Mutants into a Prototype with Human P450 Enzyme Activity
Sun-Ha Park, Chonnam National University; Dong-Hyun Kim, Chonnam National University; Chul-Ho Yun, Chonnam National University
High level expression of cytochrome P450 2C in white blood cells of mouse and rats induced by type I diabetes
Ki Tae Park, Chonnam National University; Eun Yi Cho, Chonnam National University; Taeho Ahn, Chonnam National University; Chul-Ho Yun, Chonnam National University
Interactions between Di-n-Butyl- (4-Chlorobenzohydroxamato) Tin(IV)Chloride (DBDCT) , a New Antitumor Compound with Rats Liver Cytochrome P-450
Qing-Shan Li, Shanxi Medical University; Li-Feng Zhang, Shanxi Medical University; Yao-Dong Ping, Shanxi Medical University
Confluent Growth of Huh7 Human Hepatoma Cells Induces Transcriptional Activation of the CYP3A4 Gene
Louise Sivertsson, Karolinska Institutet; Monica Ek, Karolinska Institutet; Malin Darnell, Clinical Pharmacology and DMPK; Irene Edebert, Safety Assessment, Department of Molecular Toxicology; Magnus Ingelman-Sundberg, Karolinska Institutet; Etienne P.A. Neve, Karolinska Institutet
Inter-Laboratory Evaluation Of HepaRG® Cells For Determining CYP Induction
Rebecca L. Denton, AstraZeneca R&D Charnwood; Gill Elliott, AstraZeneca R&D Charnwood; Matthew Soars, AstraZeneca R&D Charnwood; Dermot McGinnity, AstraZeneca R&D Charnwood; Arnaud M. Bruyère, Xénoblis; Françoise Brée, Xénoblis
Effect of Organic Solvents on BM3-P450 Biotransformation
Lifang Sun, Vertex Pharmaceuticals; Caroline Decker, Vertex Pharmaceuticals; Peter Grootenhuis, Vertex Pharmaceuticals; John Saunders, Vertex Pharmaceuticals; Jan N. M. Commandeur, Vrije Universiteit Amsterdam; Jelle Reinen, Vrije Universiteit Amsterdam; Nico Vermeulen, Vrije Universiteit Amsterdam
a-Naphthoflavone as an inducer or the CYP1A subfamily
Mariana Flores Torres, Instituto de Investigaciones Biomedicas, UNAM
Differential gene expression of CYP3A-isoforms in equine intestines and liver
Eva Tydén, Swedish University of Agricultural Sciences; Maria Löfgren, Swedish University of Agricultural Sciences; Hans Tjälve, Swedish University of Agricultural Sciences; Pia Larsson, Swedish University of Agricultural Sciences
Improved Predictions of Selective Estrogen Receptor Modulator and Glucocorticoid Metabolism by CYP3A4/5/7 Enzymes using Integrated Computational Models
Kiumars Shahrokh, University of Utah; Chad D. Moore, University Of Utah; Thomas E. Cheatham III, University of Utah; Garold S. Yost, University of Utah
Characterization of CYP106A1 genetic variants from various Bacillus megaterium strains
Ga-Young Lee, Chonnam National University; Chul-Ho Yun, Chonnam National University
Oriented Attachment of Cytochrome P450 Enzymes on Electrodes: Implications for Biosensor Development
Elizabeth Schneider, University of California Berkeley; Douglas S. Clark, UC Berkeley
Characteristic of Bacillus megaterium cytochrome P450 variants
Seon-Ju Choi, Chonnam National University; Chul-Ho Yun, Chonnam National University
 
9th International ISSX Meeting-Poster Presentations PDF Yazdır
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9th International ISSX Meeting-Poster Presentations

Poster Presentations

 
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