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Ana Sayfa Yağlar Enzimler Mineraller Proteinler Vitaminler Nükleik Asitler Karbonhidratlar Hormonlar Temel Biyokimya Makaleler

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Ana Sayfa
Genomics/Metabonomics/Proteomics PDF Yazdır
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Genomics/Metabonomics/Proteomics

P228
Cocaine and Amphetamine Regulated Transcript (CART) blood levels increase after Risperidon treatment in psychotic disorder patients
Tulin Yanik, MIDDLE EAST TECHNICAL UNIVERSITY; Canan Kursungoz, MIDDLE EAST TECHNICAL UNIVERSITY; Levent Sutcigil, GULHANE MILITARY MEDICAL SCHOOL; Fuat Ozgen, GULHANE MILITARY MEDICAL SCHOOL
P229
Integrated mass spectrometry based metabolomics for the biomarker discovery on the hepatotoxicity induced by carbon tetrachloride, acetaminophen and methotrexate
Byung Hwa Jung, Korea Institute of Science and Technology; Bhowmik Salil Kumar, Korea Institute of Science and Technology; Oh Seoung Kwon, Korea Institute of Science and Technology; Bong Chul Chung, Korea Institute of Science and Technology
P230
Investigating of oral constraceptives effects on weight gaining mechanisms in polycystic ovary sendrome (PCOS) patients
Tulin Yanik, MIDDLE EAST TECHNICAL UNIVERSITY; Deniz Sezlev, Middle East Technical University; Bulent Okan Yildiz, Hacettepe University
P231
Prediction of Drug-induced Liver Injury in Humans by Using Chimeric PXB-mice® with Highly Humanized Liver
Shin-Ichiro Nagatsuka, Sekisui Medical Co., Ltd.; Darina Hynes, Sekisui Medical Co., Ltd.; Shin-Ichi Ninomiya, Sekisui Medical Co., Ltd.; Masakazu Kakuni, PhoenixBio Co., Ltd.; Chise Tateno, PhoenixBio Co., Ltd.; Takashi Shimada, PhoenixBio Co., Ltd.; Yasushi Yamazoe, Tohoku University
P232
Profiling in vivo and in vitro PPARγ-mediated gene expression changes to monitor for adverse thiazolidinedione-related side effects
Jonathan M. Maher, Abbott Laboratories; Wayne R. Buck, Abbott Laboratories; Keith F. McDaniel, Abbott Laboratories; Dale J. Kempf, Abbott Laboratories; Timothy R. Middleton, Abbott Laboratories; Kevin A. Kurtz, Abbott Laboratories; Michael J. Liguori, Abbott Laboratories; Tatiana Sharapova, Abbott Laboratories; Rita X. Ciurlionis, Abbott Laboratories; Eric A. Blomme, Abbott Laboratories; Yi Yang, Abbott Laboratories
P234
The Chemotherapeutic DRUGS at the Metronomic Doses Decrease Vascular ENDOTHELIAL GROWTH FACTOR (VEGF) Secretion of SOLID TUMORS
Hande E. Aktas, Ankara University Institute of Biotechnology; Hakan Akbulut, Ankara University School of Medicine; Nalan Akgun, Ankara University School of Medicine
P235
Xenobiotic Metabolizing Enzyme Polymorphisms in a Turkish Population
Ahmet Oguz Ada, Ankara University, Faculty of Pharmacy; Volkan Karacaoglan, Ankara University, Faculty of Pharmacy; Semih C. Kunak, Giresun University, Medical Faculty; Emre Soydas, Ankara University, Faculty of Pharmacy; Mumtaz Iscan, Ankara University, Faculty of Pharmacy
 
In vitro techniques PDF Yazdır
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In vitro techniques

P285
Real-Time and Label-Free Monitoring of Bioenergetics and Cell Impedance/Adhesion for Long and Short Term Cell-Based Functional Assays in Vitro
Josef Unger, Bionas; Sabine Drechsler, Bionas; Axel Kob, Bionas; Marcus Wego, Bionas; Ralf Ehret, Bionas; Stefanie Ortinau, Bionas
P286
Isolation of Zebrafish (Danio rerio) Liver Microsomes: Protocol and Considerations
Hui Ting Chng, National University of Singapore; Han Kiat Ho, National University of Singapore; Siew Hong Lam, National University of Singapore; Eric Chun Yong Chan, National University of Singapore
P287
Oligomerization of the UGT2B7 wild-type and its mutants: homo- and heterodimerization analysis by fluorescence resonance energy transfer(FRET)
Lingmin Yuan, Zhejiang University; Lushan Yu, Zhejiang University; Su Zeng, Zhejiang University
P288
Development of A Novel Culture Plate for 3-Dimentional Cell Culture Aimed for Drug Discovery Screening
Yoko Ejiri, Kuraray Co., Ltd.; Masuhiro Nishimura, Otsuka Pharmaceutical Factory, Inc.; Masaya Hosoda, Kuraray Co., Ltd.; Motohiro Fukuda, Kuraray Co., Ltd.; Shinsaku Naito, Otsuka Pharmaceutical Factory, Inc.
P289
Induced Expressions and Activities of Drug-Metabolizing Enzymes in the Human Hepatocellular Carcinoma Cell Line Cultured On the Micro-Space Cell Culture Plates
Akane Yoshida, Chiba University; Kaoru Kobayashi, Chiba University; Yoko Ejiri, Kuraray Co., Ltd.; Sachiko Takagi, Chiba University; Hanaka Mimura, Chiba University; Masaya Hosoda, Kuraray Co., Ltd.; Kan Chiba, Chiba University
P290
Assessment of a human in vitro system as an alternative for S-9 fraction to predict in vivo metabolic profiles for drugs
Amin Kamel, Novartis Institutes for BioMedical Research; Mithat Gunduz, Novartis Institutes for BioMedical Research; Kevin Colizza, Novartis Institutes for BioMedical Research; Franco Lombardo, Novartis Institutes for BioMedical Research; Shawn Harriman, Novartis Institutes for BioMedical Research
P291
Characterization of the Tight Junction Integrity in Different Renal Cell Cultures
Christian Lechner, Bayer Schering Pharma AG; Gert Fricker, Heidelberg University; Andrea Thiele, Bayer Schering Pharma AG; Andreas Reichel, Bayer Schering Pharma AG; Ursula Moenning, Bayer Schering Pharma AG
P292
Microsomal Protein Binding in IVIVE
Alison Meechan, Charles River; Lisa McBride, Charles River; Jon Welch, Charles River; Fiona Milligan, Charles River; Stephen Madden, Charles River
P294
Vinorelbine's effects on the cell cycle progression in HeLa cell line
Ozlem Gokce, Faculty of Medicine, Gazi University; Akin Yilmaz, Faculty of Medicine, Gazi University; Venhar Gurbuz, Faculty of Medicine, Gazi University; Ece Konac, Faculty of Medicine, Gazi University; Abdullah Ekmekci, Faculty of Medicine, Gazi University
P295
Apoptotic effects of cisplatin on human colon cancer cell line (HT29)
Venhar Gurbuz, Faculty of Medicine, Gazi University; Akin Yilmaz, Faculty of Medicine, Gazi University; Ozlem Gokce, Faculty of Medicine, Gazi University; Ece Konac, Faculty of Medicine, Gazi University
 
Herbal Medicine-Active Compounds PDF Yazdır
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Herbal Medicine-Active Compounds

P250
Dimethyl-Diphenyl-Bicarboxylate (DDB) as Antiapoptotic Agent Targeting Death Ligand and Caspases Signaling Pathway in a Model of Hepatic Ischemia Reperfusion Injury
Alshaymaa Amin El-Bahy, The German university in Cairo
P248
Aldose reductase natural inhibitors from ethyl acetate extracts from southern Turkey
Melih Onay, Middle East Technical University; Nursen Coruh, Middle East Technical University; Belgin İşgör, Atılım University
P256
Phenethyl Isothiocyanate and Sulforaphane Mediated Apoptotic Cell Death in Human Prostate Cancer Cells Is Initiated by Mitochondria Generated Reactive Oxygen Species
Shivendra Vikram Singh, Univ of Pittsburgh Cancer Inst; Dong Xiao, Univ of Pittsburgh Cancer Inst; Anna A Powolny, Univ of Pittsburgh Cancer Inst; Su-Hyeong Kim, Univ of Pittsburgh Cancer Inst; Eun-Ryeong Hahm, Univ of Pittsburgh Cancer Inst
P252
Evaluation of selected herbal remedies sold in Libyan market for treatment of diabetes
Mukhtar R. Haman, Faculty of Pharmacy, AlFateh University
P254
Living knowledge of the healing plants: ethno-phytotherapy in the Local people, Santal and Orao ethnic groups from the Rangpur district of Bangladesh
Md. Ariful Haque Mollik, Peoples Integrated Alliance
P257
Plasma Pharmacokinetics and Urinary Excretion of Ginsenosides after Oral Administration of Panax notoginseng Extract to Human Subjects
Feifei Du, Shanghai Institute of Materia Medica; Fang Xu, Shanghai Institute of Materia Medica; Chuan Li, Shanghai Instiyute of Materia Medica
P249
Dietary Aromatase Inhibitors in Human Non–Small Cell Lung Cancer
Alaattin Sen, Pamukkale University; Hakan Akca, Pamukkale University; Gurbet Celik, Pamukkale University
P253
Ginger consitutents modulate function and expression of p-gp and bcrp
Sabrina Nickel, Heidelberg University; Anne Mahringer, Heidelberg University; Gert Fricker, Heidelberg University; Valeska Reichel, Heidelberg University
P251
Effects of Avaricon® on High Fat Diet-induced Hepatosteatosis, Oxidative Stress and Lipid Profile in Rats
Jelena Calasan, Faculty of Medicine; Vesna Mijatovic, Faculty of Medicine; Biljana Bozin, Faculty of Medicine; Isidora Samojlik, Faculty of Medicine; Olga Horvat, Faculty of Medicine
P255
Natural resveratrol analogs arachidin-1, arachidin-3 and piceatannol bind human and mice cannabinoid receptors CB1 and CB2
Paul L. Prather, University of Arkansas for Medical Sciences; Lisa K. Cortez, University of Arkansas for Medical Sciences; Luis Nopo-Olazabal, Arkansas State University; Vipin Nair, Arkansas State University; Fabricio Medina-Bolivar, Arkansas State University; Anna Radominska-Pandya, University of Arkansas for Medical Sciences
P258
Prooxidant and Antioxidant Effects of Three Dietary Flavonoids and Their Mixtures
Burcu Eren, Ege University, Faculty of Pharmacy; Hande Gurer-Orhan, Ege University, Faculty of Pharmacy
 
Mechanisms of xenobiotic toxicities PDF Yazdır
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Mechanisms of xenobiotic toxicities

Cyclopiazonic acid toxic effects on the liver and kidneys: biochemical and histopathological studies
Hassan Malekinejad, Urmia University; Peyman Akbari, Urmia University
Attenuation of Neurotoxicity Induced by Sub-Chronic Paraquat Administration in Rats by Deprenyl, Quercetin, Green Tea or Malt Extract
Nesrine Salah El Dine El Sayed, Lecturer of Pharmacology & Toxicology; Hala Fahmy Zaki, Associate professor of Pharmacology & Toxicology
Association of blood level of methemoglobin with clinical outcome of patients with aluminium phosphide poisoning
Babak Mostafazadeh, Shaheed Beheshty University Of Medical Sciences; Esmaeil Farzaneh, Ardabil University Of Medical Sciences; Tahmineh Afsharian, Private Physician
Benefit Effect of Naloxone in Benzodiazepines Intoxication:Findings of a Preliminary Study
Babak Mostafazadeh, Shaheed Beheshty University Of Medical Sciences; Esmaeil Farzaneh, Ardabil University Of Medical Sciences; Tahmineh Afsharian, Private Physician
Effect of Exposure to Bile Salts on Urea Formation in Sandwich-Cultured Rat Hepatocytes
Sagnik Chatterjee, Katholieke Universiteit Leuven; Patrick Augustijns, Katholieke Universiteit Leuven; Pieter Annaert, Katholieke Universiteit Leuven
Transcriptomics analysis of the Artemisinin stress response in mouse embryonic stem cells
M. Raamsman-Ossevoort, Leiden University, Leiden/Amsterdam Center for Drug Research; J. Carreras Puigvert, Leiden University, Leiden/Amsterdam Center for Drug Research; B. Van de Water, Leiden University, Leiden/Amsterdam Center for Drug Research
Deuterium insertion approach to reduce metabolism-mediated liabilities: Integration of biotransformation results and structural modification into potential toxicity findings
Amin Kamel, Novartis Institutes for BioMedical Research; Mithat Gunduz, Novartis Institutes for BioMedical Research; Natalie Dales, Novartis Institutes for BioMedical Research; Clayton Springer, Novartis Institutes for BioMedical Research; Suzie Ferreira, Novartis Institutes for BioMedical Research; Franco Lombardo, Novartis Institutes for BioMedical Research; Shawn Harriman, Novartis Institutes for BioMedical Research
TNF-alpha enhances cisplatin-induced renal injury via the JNK and NF-kB pathways
Giulia O.E. Benedetti, Lacdr; J. Meerman, Lacdr; B. van de Water, Lacdr; M. de Graauw, Lacdr
Metabolic Activation of Chlorogenic Acid in vitro and in vivo
Xiaoyan Chen, Shanghai Institute of Materia Medica, Chinese Academy of Sciences; Cen Xie, Shanghai Institute of Materia Medica, Chinese Academy of Sciences; Tao Yuan, Shanghai Institute of Materia Medica, Chinese Academy of Sciences; Dafang Zhong, Shanghai Institute of Materia Medica, Chinese Academy of Sciences
Precision-cut liver slices as an ex vivo model to study idiosyncratic hepatotoxicity in mouse and human
Mackenzie Hadi, University of Groningen; Yixi Chen, University of Groningen; Harry Emmen, NOTOX B.V.; Miranda Stitzinger, NOTOX B.V.; Geny Groothuis, University of Groningen
Erdosteine has dual effects on haemostasis via its different metabolites in young rats
Süleyman Oktar, Medical Faculty of Mustafa Kemal University; Vefik Arica, Medical Faculty of Mustafa Kemal University; Murat Tutanc, Medical Faculty of Mustafa Kemal University; Oktay Hasan Ozturk, Medical Faculty of Mustafa Kemal University
Acute disruption of bone marrow hematopoietic progenitor cells by benzo(a)pyrene (BP) is reversed by processes dependent on Ah Receptor activation
Alhaji U. N'Jai, University of Wisconsin Madison; Michele Larsen, University of Wisconsin Madison; Charles J. Czuprynski, University of Wisconsin Madison; Colin R. Jefcoate, University of Wisconsin Madison
Mechanism of Hepatoprotective Effect of Tamoxifen Against Drug-induced Liver Injury
Tsuyoshi Yokoi, Faculty of Pharmaceutical Sciences, Kanazawa University; Yukitaka Yoshikawa, Faculty of Pharmaceutical Sciences, Kanazawa University; Yasuyuki Toyoda, Faculty of Pharmaceutical Sciences, Kanazawa University; Satonori Higuchi, Faculty of Pharmaceutical Sciences, Kanazawa University; Tohru Tsukui, Research Center for Genomic Medicine; Koichi Tsuneyama, Department of Diagnostic Pathology; Tatsuki Fukami, Faculty of Pharmaceutical Sciences, Kanazawa University; Miki Nakajima, Faculty of Pharmaceutical Sciences, Kanazawa University
Exploiting the Third Dimension for Predicting Drug Induced in vitro Nephrotoxicity
Sreenivasa Ramaiahgari, Leiden University; Bob van de Water, LACDR, Leiden University; Leo Price, Leiden University
Influence of valproate on the levels of tri- and diphosphate nucleotides in rat liver tissues
Paula B. M. Luis, Faculdade de Farmácia, Universidade de Lisboa; Lodewijk IJlst, Laboratory Genetic Metabolic Diseases, Dep. Clinical Chemistry and Pediatrics, AMC, University of Amsterdam, The Netherlands; Jeroen Roelofsen, Amsterdam Medical Centre, University of Amsterdam; André B.P. van Kuilenburg, Amsterdam Medical Centre, University of Amsterdam; Marinus Duran, Laboratory Genetic Metabolic Diseases, Dep. Clinical Chemistry and Pediatrics, AMC, University of Amsterdam, The Netherlands; Isabel Tavares de Almeida, Faculdade de Farmácia, Universidade de Lisboa; Ronald J.A. Wanders, Laboratory Genetic Metabolic Diseases, Dep. Clinical Chemistry and Pediatrics, AMC, University of Amsterdam, The Netherlands; Margarida F.B. Silva, Faculdade de Farmácia, Universidade de Lisboa
Evidences of covalent adduct formation of quinoline compounds and their phase I metabolites with glutathione and N-acetyl cysteine
Bhagwat Prasad, National Institute of Pharmaceutical Education and Research (NIPER), SAS Nagar 160062, Punjab, India; Amit Garg, National Institute of Pharmaceutical Education and Research (NIPER), SAS Nagar 160062, Punjab, India; Saranjit Singh, National Institute of Pharmaceutical Education and Research (NIPER), SAS Nagar 160062, Punjab, India; Rahul Jain, National Institute of Pharmaceutical Education and Research (NIPER), SAS Nagar 160062, Punjab, India
Effect of Phenobarbital on the Cytotoxicity of Valproic Acid and 2-Ene-Valproic Acid in Sandwich Cultures of Rat Hepatocytes
Jayakumar Surendradoss, Univ of British Columbia; Stoyan Karagiozov, Univ of British Columbia; Thomas K. H. Chang, Univ of British Columbia; Frank S. Abbott, Univ of British Columbia
Potential biomarker for the assessment of hepatotoxicity induced by metabolic activation of pyrrolizidine alkaloids
Ge Lin, The Chinese University of Hong Kong; Na Li, The Chinese University of Hong Kong; Mi Li, The Chinese University of Hong Kong; Wood-Yee Chan, The Chinese University of Hong Kong; Peter P. Fu, National Center for Toxicological Research; Hong-Xi Xu, Hong Kong Jockey Club Institute of Chinese Medicine
 
Risk Assessment PDF Yazdır
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Risk Assessment

P447
Assessment of Sodium Dodecyl Sulfate-Induced Irritation on a Preclinical Model of Pig Ear Skin Organ Culture
Daniel Bacqueville, Centre de Recherche et Développement Pierre Fabre Dermo-Cosmétique; Valérie Ortis, Centre de Recherche et Développement Pierre Fabre Dermo-Cosmétique; Anne-Sophie Jimenez, Centre de Recherche et Développement Pierre Fabre Dermo-Cosmétique; Marie Boisson, Centre de Recherche et Développement Pierre Fabre Dermo-Cosmétique; Hélène Duplan, Centre de Recherche et Développement Pierre Fabre Dermo-Cosmétique
P453
Semi-quantitative assessment of reactive metabolite formation of 60 marketed drugs using the bi-functional trapping reagent dansyl-γGlu-Cys-Lys
Ralf Schmidt, AstraZeneca R&D Montreal; Rosemarie Panetta, AstraZeneca R&D Montreal
P450
Investigation into the incidence of control sample contamination in toxicokinetic samples generated during regulatory toxicology studies
Robert G. Turcan, Covance Labs Inc; Sarah Cahill, Covance Labs Inc
P449
Gene Profiling of Drug-metabolizing Enzymes in Normal Human Bronchial Epithelial Cells Exposed to Single-walled Carbon Nanotubes
Kotaro Hitoshi, Meijo University; Miki Katoh, Meijo University; Tomoko Suzuki, Meijo University; Yoshinori Ando, Meijo University; Masayuki Nadai, Meijo University
P448
Covalent Binding of Drug Candidates to Proteins as a Reactive Metabolite Risk Assessment Tool
Emre M. Isin, AstraZeneca R&D Mölndal; Jesper Nilsson, AstraZeneca R&D Mölndal; Johanna Midlöv, AstraZeneca R&D Mölndal; Göran N. Nilsson, AstraZeneca R&D Mölndal; Carina Leandersson, AstraZeneca R&D Mölndal; Richard A. Thompson, AstraZeneca R&D Mölndal
P451
Methylation markers of arsenic associated urothelial carcinoma in peripheral blood leukocyte
Tse-Yen Yang, National Defense Medical Center; Ling-I Hsu, Academia Sinica; Chien-Jen Chen, Academia Sinica
P452
Occurrence of ochratoxin A in various food products in Turkey
Buket Alpertunga, Faculty of Pharmacy, Istanbul University; Sibel Ozden, Faculty of Pharmacy, Istanbul University; Ayse Sibel Akdeniz, Faculty of Pharmacy, Istanbul University
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